Tirzepatide is an innovative dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist designed for treating type 2 diabetes, obesity, and associated metabolic disorders. Its unique dual agonist mechanism enables superior metabolic control, significant weight reduction, and comprehensive improvements in glycemic management. While not yet FDA-approved for general therapeutic use, extensive clinical trials strongly support its remarkable therapeutic potential.